Posted on July 30, 2008 by crimsoncanary
J&J have published a series of Aurora A/VEGFR-2 inhibitors
Filed under: kinase | Tagged: Aurora A, J&J, Johnson and Johnson, kinase, VEGFR-2, VEGFR2 | Comments Off
Posted on July 30, 2008 by crimsoncanary
AstraZeneca have published a series of pyridyl and thiazolyl bisamide CSF-1R inhibitors for the treatment of cancer
Filed under: Kinase receptor | Tagged: AstraZeneca, CSF-1R, CSF1R, Preclinical, Research | Comments Off
Posted on July 30, 2008 by crimsoncanary
Amgen have published a series of Indazole KDR/VEGFR-2 Inhibitors
Filed under: kinase | Tagged: Amgen, KDR, kinase, VEGFR-2, VEGFR2 | Comments Off
Posted on July 30, 2008 by crimsoncanary
In 2nd quarter results Incyte have provided an update on JAK2 inhibitors INC18424 and INCB28050
Filed under: kinase | Tagged: INCB-18424, INCB-28050, INCB18424, INCB28050, Incyte, JAK, JAK2, kinase | Comments Off
Posted on July 30, 2008 by crimsoncanary
ARIAD have announced the initiation of a Phase II clinical trial of mTOR inhibitor Deforolimus in Patients with Metastatic, HER2-Positive Breast Cancer
Filed under: kinase | Tagged: AP-23573, AP23573, Ariad, deforolimus, kinase, Merck, MK-8669, MK8669, mTOR, Phase II | Comments Off
Posted on July 30, 2008 by crimsoncanary
Novartis have published a series of 4-(1H-Indazol-5-yl)-6-phenylpyrimidin-2(1H)-one analogs as potent CDC7 inhibitors
Filed under: kinase | Tagged: cdc7, kinase, Novartis, Preclinical, Research | Comments Off